Theophylline

Buy Theophylline
theophylline

$23.70

  • Active ingredient: Theophylline
  • Category: Allergy & Asthma
  • Delivery time: Airmail (14-21 days) | EMS trackable (5-9 days)
  • Prescription: Included
  • Availability: In Stock

Theophylline 400mg pills are available to order from our licensed Malaysian pharmacy. This medication functions as a phosphodiesterase inhibitor and a non-selective adenosine receptor antagonist, leading to the relaxation of smooth muscles in the airways, which helps ease breathing. It serves as a long-term maintenance therapy for adults managing chronic symptoms related to persistent asthma or chronic obstructive pulmonary disease (COPD).

Table of contents

Product Information

Generic Theophylline is a long-acting bronchodilator available in pill form, commonly prescribed for Asthma and certain allergic airway conditions. Delivered through our discreet online pharmacy, it arrives in plain packaging with secure shipping throughout Malaysia. Understanding how this medication relaxes airway muscles helps patients grasp why it may be part of an asthma management plan, especially when inhaled therapies alone are insufficient.

Theophylline Overview
Active Ingredient Theophylline
Drug Class Methylxanthine bronchodilator
Primary Uses Chronic asthma, COPD exacerbation prevention, occasional severe bronchospasm
Available Forms Oral tablet
Typical Strength(s) 400 mg
Administration Swallow whole with water
Side Effects Mild: nausea, headache; Common: insomnia, tremor; Severe: cardiac arrhythmia
Onset of Action 30-60 minutes

Understanding Generic Theophylline

Generic Theophylline represents the chemical substance without brand-specific additives, confirming bioequivalence to any proprietary version. Classified as a methyl-xanthine, it is regulated as a prescription-only medication in Malaysia, ensuring physician oversight before dispensing. By offering a cost-effective alternative, patients gain access to the same therapeutic impact while reducing out-of-pocket expenses. The tablet formulation delivers a steady plasma concentration that supports long-term airway stability.

How Does Theophylline Work?

Theophylline exerts its bronchodilatory effect primarily by inhibiting phosphodiesterase-4 (PDE4), an enzyme that breaks down cyclic AMP (cAMP) inside smooth-muscle cells. Elevated cAMP levels cause the muscles surrounding the bronchi to relax, widening the airway passages and easing breathing. Additionally, the drug antagonizes adenosine receptors, reducing inflammation-related bronchoconstriction. After oral ingestion, absorption occurs within an hour, and peak plasma levels are reached by 2-3 hours. The half-life ranges from 6 to 8 hours in healthy adults but can extend in the elderly or those with liver impairment, influencing dosing intervals. Metabolism proceeds via hepatic cytochrome P450 enzymes, leading to renal excretion of metabolites. Understanding these pharmacokinetic steps clarifies why steady dosing is crucial to maintain therapeutic levels without triggering toxicity.

Clinical Applications of Theophylline

In chronic asthma, Theophylline serves as an adjunct to inhaled corticosteroids and long-acting β2-agonists, especially when patients experience persistent symptoms despite optimal inhaler use. Its smooth-muscle relaxation reduces nocturnal bronchospasm, improving sleep quality and daytime activity. For chronic obstructive pulmonary disease (COPD), the drug can lessen the frequency of exacerbations, complementing bronchodilator regimens. Occasionally, clinicians prescribe Theophylline for severe Allergic Reactions that involve bronchial hyper-responsiveness when epinephrine or antihistamines alone are insufficient. Because its therapeutic window is narrow, regular blood-level monitoring guides dose adjustments, ensuring effectiveness while avoiding adverse cardiac effects. Theophylline’s role is generally reserved for patients who need an additional oral agent to stabilize airway tone, positioning it as a second-line or maintenance option rather than first-line monotherapy.

Determining Patient Suitability

Ideal candidates for Theophylline are adults with documented asthma or COPD who continue to experience symptoms despite inhaled therapy. Patients should have normal liver function and no history of severe cardiac arrhythmias, as these conditions heighten toxicity risk. Elderly individuals often metabolize the drug more slowly, necessitating lower starting doses and closer monitoring. Pregnancy classification places Theophylline in Category C, indicating that potential benefits may outweigh risks only under medical supervision. Individuals with a known hypersensitivity to methyl-xanthines, such as caffeine or theobromine, should avoid the medication. If a patient regularly consumes high-caffeine beverages, dose adjustments might be required because caffeine competes for the same metabolic pathway, potentially elevating plasma concentrations.

Optimizing Theophylline Dosing and Lifestyle

Consistent timing helps maintain stable blood levels; taking the tablet at the same hour each day, preferably with a meal, reduces gastrointestinal irritation and improves absorption. A light snack containing a modest amount of fat can modestly increase bioavailability, but excessive fatty meals may delay onset. Night-shift workers should coordinate dosing with their sleep schedule to avoid insomnia-a common side effect linked to the drug’s central nervous system stimulation. When traveling, store tablets in a cool, dry place away from direct sunlight; prolonged heat exposure may degrade potency. If a dose is missed, patients should take it as soon as remembered, provided it is more than six hours before the next scheduled dose; otherwise, skipping the missed pill prevents accidental double-dosing.

Monitoring Treatment Effectiveness

Physicians typically order serum Theophylline concentrations after the patient reaches a steady-state regimen, aiming for a therapeutic range of 10-20 µg/mL. Levels below 10 µg/mL may indicate suboptimal bronchodilation, while concentrations above 20 µg/mL increase the likelihood of cardiac or neurological toxicity. Routine monitoring includes checking heart rhythm, blood pressure, and signs of tremor or Agitation. Patients should report any new palpitations, dizziness, or persistent Nausea, prompting the clinician to reassess dosage or investigate drug interactions. Adjustments are made incrementally, reflecting the drug’s narrow therapeutic index and the goal of achieving symptom control with the lowest effective dose.

Managing Potential Side Effects

When Theophylline triggers nausea, the underlying mechanism often involves direct stimulation of the chemoreceptor trigger zone in the brainstem. Taking the tablet with food or a small amount of antacid can mitigate this effect. Headaches and Insomnia arise from central nervous system excitation; limiting caffeine intake and maintaining a regular sleep routine reduce their incidence. Tremors result from enhanced catecholamine release; patients may find relief by adjusting the dose downward under medical guidance. Should any severe symptom such as rapid heartbeat, chest Pain, or Seizures emerge, immediate medical attention is essential, as these indicate plasma levels entering the toxic range. Continuous communication with a healthcare provider ensures timely intervention before complications develop.

Drug Interactions and Precautions

Theophylline metabolism is highly susceptible to interference from other medications. Agents that inhibit cytochrome P450-such as Erythromycin, Ciprofloxacin, and certain antifungals-can raise Theophylline concentrations, heightening toxicity risk. Conversely, enzyme inducers like rifampin, carbamazepine, or smoking (which increases hepatic clearance) may lower drug levels, reducing efficacy. Patients should disclose all prescriptions, over-the-counter products, and herbal supplements to their physician. Alcohol consumption amplifies central nervous system effects and may precipitate gastric irritation; moderate intake is advisable. Adjusting doses when starting or stopping interacting drugs helps maintain therapeutic balance.

Accessing Theophylline Through Our Service

Obtaining Generic Theophylline begins with a valid prescription from a licensed Malaysian physician. Once the prescription is uploaded to our platform, our pharmacy team verifies the details and prepares the medication for discreet shipment. The ordering process is fully digital, allowing patients to track delivery status in real time. Competitive pricing reflects bulk purchasing power, delivering savings compared with traditional brick-and-mortar pharmacies. By choosing our service, patients benefit from convenient home delivery, secure packaging, and personalized support for any questions about dosing or side-effect management.


Frequently Asked Questions

Can I take Theophylline with my inhaler?

Yes, Theophylline is intended to complement inhaled bronchodilators, not replace them. Using both agents can improve overall airway control, especially during nighttime symptoms.

How soon will I feel relief after the first dose?

Most individuals notice a reduction in wheezing and shortness of breath within 30-60 minutes, as the drug begins to relax bronchial muscles and raise cAMP levels.

Is it safe to consume coffee while on Theophylline?

Both substances share the methyl-xanthine pathway, so high caffeine intake may increase plasma Theophylline concentrations. Limiting coffee to one small cup per day is generally advisable.

What should I do if I miss a dose?

Take the missed tablet as soon as you remember, unless the next scheduled dose is less than six hours away; in that case, skip the missed dose and continue with the regular schedule.

Can Theophylline be used in children?

Pediatric use is possible but requires careful dosing based on weight and close serum level monitoring. Only a pediatrician can prescribe it for minors.

Will Theophylline affect my ability to drive?

Mild Sedation or tremor can occur, especially at higher concentrations. If you feel unusually drowsy or shaky, avoid operating vehicles until you know how the medication affects you.

How often must my blood levels be checked?

Initial monitoring occurs after five to seven days of steady dosing. Subsequent checks are typically performed whenever the dose changes, new interacting drugs are added, or symptoms suggest toxicity.

Is Theophylline covered by Malaysian health insurance?

Coverage varies by plan. Some private insurers include oral asthma medications, while public schemes may limit reimbursement. Verify with your provider before ordering.

Why does my heart race after taking Theophylline?

Elevated cAMP not only relaxes airway muscles but also increases cardiac contractility and conduction speed, which can manifest as palpitations if blood levels rise too high.

Can I travel internationally with my medication?

Yes, as long as you carry a copy of the prescription and keep the tablets in their original packaging. Declare the medication at customs if required by the destination country.


Glossary

Bronchodilator
A drug that relaxes the muscles of the airways, widening them to improve airflow.
cAMP (Cyclic Adenosine Monophosphate)
A cellular messenger that, when increased, leads to smooth-muscle relaxation in the lungs.
Therapeutic window
The range of drug concentrations in the blood that provides benefit without causing harmful side effects.
Cytochrome P450
A group of liver enzymes responsible for metabolizing many medications, including Theophylline.
Bioequivalence
When a generic drug delivers the same amount of active ingredient to the bloodstream as the brand-name version.

Important Information

The content presented here offers general knowledge about Generic Theophylline and does not replace professional medical advice. Use of this medication should be guided by a qualified healthcare provider, who can assess individual risks, monitor blood levels, and adjust dosing as needed. Off-label applications are not endorsed without physician supervision. Our pharmacy service facilitates convenient access and potential cost savings, but final responsibility for safe use rests with the patient and their prescriber. Always read the prescription label and consult your doctor with any concerns.


How to Buy Theophylline Online in Malaysia


Is Theophylline Available in Malaysia?

Theophylline is available in Malaysia without a prescription from our online pharmacy. We source products from verified international suppliers in bulk and comply fully with Malaysian import regulations. Personal-use orders do not require a local prescription.

Steps to Buy Theophylline Legally and Affordably in Malaysia

Ordering Theophylline through our pharmacy is simple. Select the required dosage and quantity, add it to your cart, and proceed to checkout—or continue adding more medications before finalizing your order. A prescription is not required on your part, as our overseas trading partner will issue it for you. This ensures that your medication arrives directly at your doorstep, discreetly packaged and fully compliant with local regulations. The process is efficient, safe, and hassle-free.

Can I Import Theophylline into Malaysia?

Importing Theophylline into Malaysia for personal use is allowed under local guidelines. Our pharmacy ensures that all orders meet the necessary criteria, including valid prescriptions issued overseas and approved quantities. You can choose from trusted generic alternatives or affordable branded versions.

Tips for Save Money on Theophylline in Malaysia

  • Opt for generic alternatives like Theophylline for the same therapeutic effects at a lower price.
  • Compare prices and choose our pharmacy for fair rates and quality assurance.
  • Take advantage of special discounts and additional savings available through our platform.

Refilling Your Theophylline Prescription in Malaysia

Refilling your prescription with us is quick and convenient. By using your account, you can enjoy exclusive discounts of 10% on every refill, making your treatment plan even more affordable. Our user-friendly platform ensures you can reorder with ease whenever needed.

Reasons Customers Choose Us

Our service is designed to meet the needs of customers in Malaysia. We comply with all local import regulations, ensuring safe and prompt delivery across the country. With shipping options covering major cities like Kuala Lumpur, Johor Bahru, Penang, and more, we provide timely and discreet service. We also place strong emphasis on privacy, ensuring maximum protection of your personal information. Our quality assurance process guarantees high-quality medications, and we offer wide delivery coverage across Asia so that you can access your treatments wherever you are. Trust us for quality medications, exceptional privacy standards, and personalized support every step of the way.


Theophylline Drug Class

Methylxanthines

Theophylline Connected Conditions

How to purchase Theophylline on our Online Drugstore

To purchase Theophylline on our website, just select the required dosage and quantity of pills above. The price of your choice will appear automatically. Next, add the chosen amount to your cart by clicking the Add to Cart button. You can either continue shopping for more pills or proceed to the checkout. At the Checkout, finalize your purchase through our secure payment gateway, which supports Malaysian customers.

Theophylline / Theophylline pills are made using high-quality generic ingredients and manufactured under strict quality control in accordance with WHO and National Pharmaceutical Regulatory Agency (NPRA) standards. Please note that Theophylline pills are shipped from overseas, as prescriptions are issued outside of Malaysia to ensure compliance with international import guidelines.

Disclaimer

The content on this website is provided for informational purposes only and is not intended to replace professional medical advice, diagnosis, or treatment. Always consult a licensed doctor, pharmacist, or healthcare provider in Malaysia for any questions regarding your health or medication. Do not ignore or delay seeking medical advice based on information found here. Use of this website does not establish a doctor-patient relationship. In the event of a medical emergency in Malaysia, please call the national emergency number 999 or visit the nearest hospital or clinic immediately. This website and its operators assume no responsibility or liability for any errors, omissions, or outcomes arising from the use of the information provided.

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Theophylline

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